Imiloxan is a drug which is used in scientific research.
It acts as a selective antagonist for the α2B adrenergic receptor,[1] and has been useful for distinguishing the actions of the different α2 adrenergic subtypes.
[2][3] The imidazole portion of imiloxan is prepared by the reaction of an imidate with the diethyl acetal of aminoacetaldehyde.
N-Alkylation of the imidazole with ethyl iodide gives imiloxan.
This antihypertensive-related article is a stub.