[5][6][7] This gene encodes a protein that functions in genome maintenance (double strand break repair).
[15] Variants in the PALB2 gene are associated with an increased risk of developing breast cancer [16] of magnitude similar to that associated with BRCA2 mutations [17] and PALB2-deficient cells are sensitive to PARP inhibitors.
[7] Mutations in this gene have been associated with an increased risk of ovarian, breast and pancreatic cancer.
[24] This reduced fertility appears to be due to germ cell attrition resulting from a combination of unrepaired DNA breaks during meiosis and defective synapsis of the X and Y chromosomes.
[citation needed] The PALB2-BRCA1 interaction is likely important for repairing such damages during male meiosis.
Characterized domaines of PALB2
Recombinational repair of DNA double-strand damage - some key steps.
ATM
(ATM) is a
protein kinase
that is recruited and activated by
DNA double-strand breaks
. DNA double-strand damages also activate the
Fanconi anemia core complex
(FANCA/B/C/E/F/G/L/M).
[
8
]
The FA core complex
monoubiquitinates
the downstream targets FANCD2 and FANCI.
[
9
]
ATM activates (phosphorylates)
CHEK2
and FANCD2
[
10
]
CHEK2 phosphorylates BRCA1.
[
11
]
Ubiquinated FANCD2 complexes with
BRCA1
and
RAD51
.
[
12
]
The PALB2 protein acts as a hub,
[
13
]
bringing together BRCA1, BRCA2 and RAD51 at the site of a DNA double-strand break, and also binds to RAD51C, a member of the RAD51 paralog complex
RAD51B
-
RAD51C
-
RAD51D
-
XRCC2
(BCDX2). The BCDX2 complex is responsible for RAD51 recruitment or stabilization at damage sites.
[
14
]
RAD51
plays a major role in
homologous recombinational
repair of DNA during double strand break repair. In this process, an ATP dependent DNA strand exchange takes place in which a single strand invades base-paired strands of homologous DNA molecules. RAD51 is involved in the search for homology and strand pairing stages of the process.